PubMed:pH oscillations and mechanistic analysis in the hydrogen peroxide-sulfite-thiourea reaction system. |
PubMed:Cerium(III/IV) formamidinate chemistry, and a stable cerium(IV) diolate. |
PubMed:Probing the limits of ligand steric bulk: backbone C-H activation in a saturated N-heterocyclic carbene. |
PubMed:Topical treatment with probiotic Lactobacillus brevis CD2 inhibits experimental periodontal inflammation and bone loss. |
PubMed:Concerted halogen bonding and orthogonal metal-halogen interactions in dimers of lithium formamidinate and halogenated formamidines: an ab initio study. |
PubMed:New azido-substituted tantalum compounds: syntheses and DFT examination of nitrogen-rich mono-, di-, and trinuclear tantalum(V) compounds. |
PubMed:Acaricide and ivermectin resistance in a field population of Rhipicephalus microplus (Acari: Ixodidae) collected from red deer (Cervus elaphus) in the Mexican tropics. |
PubMed:The protective effect of HET0016 on brain edema and blood-brain barrier dysfunction after cerebral ischemia/reperfusion. |
PubMed:In vitro induction of apoptosis and necrosis by new derivatives of daunorubicin. |
PubMed:Amitraz. |
PubMed:Competition between hydrogen bonds and halogen bonds in complexes of formamidine and hypohalous acids. |
PubMed:In vitro and in vivo evaluation of cypermethrin, amitraz, and piperonyl butoxide mixtures for the control of resistant Rhipicephalus (Boophilus) microplus (Acari: Ixodidae) in the Mexican tropics. |
PubMed:Synthesis, structure, and reactivity of lanthanide complexes incorporating indolyl ligands in novel hapticities. |
PubMed:20-Hydroxyeicosatetraenoic acid inhibition attenuates balloon injury-induced neointima formation and vascular remodeling in rat carotid arteries. |
PubMed:Increased 20-HETE synthesis explains reduced cerebral blood flow but not impaired neurovascular coupling after cortical spreading depression in rat cerebral cortex. |
PubMed:Evaluation of the DNA damaging effects of amitraz on human lymphocytes in the Comet assay. |
PubMed:Selective oxidation of thiourea with H(2)O(2) catalyzed by [Ru(III)(edta)(H(2)O)](-): kinetic and mechanistic studies. |
PubMed:Synergistic actions of formamidine insecticides on the activity of pyrethroids and neonicotinoids against Aedes aegypti (Diptera: Culicidae). |
PubMed:Unique stepwise substitution reaction of a mono(guanidinate)tetraplatinum complex with amidines, giving mono(amidinate)tetraplatinum complexes through mixed-ligand intermediate complexes. |
PubMed:Synthesis, structures and reactivity of lanthanoid(II) formamidinates of varying steric bulk. |
PubMed:Treatment with the cytochrome P450 ω-hydroxylase inhibitor HET0016 attenuates cerebrovascular inflammation, oxidative stress and improves vasomotor function in spontaneously hypertensive rats. |
PubMed:Molecular cloning and pharmacological characterisation of a tyramine receptor from the rice stem borer, Chilo suppressalis (Walker). |
PubMed:Thermal fluctuations and infrared spectra of the formamide-formamidine complex. |
PubMed:Synthesis of biologically active and photostable rigid poly(vinyl chloride). |
PubMed:20-HETE induces hyperglycemia through the cAMP/PKA-PhK-GP pathway. |
PubMed:Chronic doxorubicin cardiotoxicity modulates cardiac cytochrome P450-mediated arachidonic acid metabolism in rats. |
PubMed:Increased expression of CYP4Z1 promotes tumor angiogenesis and growth in human breast cancer. |
PubMed:Analogs of N'-hydroxy-N-(4H,5H-naphtho[1,2-d]thiazol-2-yl)methanimidamide inhibit Mycobacterium tuberculosis methionine aminopeptidases. |
PubMed:Amitraz poisoning. |
PubMed:Inhibitors of 20-hydroxyeicosatetraenoic acid (20-HETE) formation attenuate the natriuretic effect of dopamine. |
PubMed:Nitrogen incorporation in CH(4)-N(2) photochemical aerosol produced by far ultraviolet irradiation. |
PubMed:Sodium chloride concentration affects yield, quality, and sensory acceptability of vacuum-tumbled marinated broiler breast fillets. |
PubMed:Protective effect of 20-hydroxyeicosatetraenoic acid (20-HETE) on adriamycin-induced toxicity of human renal tubular epithelial cell (HK-2). |
PubMed:Assessment of the adverse effects of the acaricide amitraz: in vitro evaluation of genotoxicity. |
PubMed:Attenuation of neonatal ischemic brain damage using a 20-HETE synthesis inhibitor. |
PubMed:Protective effect of 20-HETE inhibition in a model of oxygen-glucose deprivation in hippocampal slice cultures. |
PubMed:Evidence for a common pharmacological interaction site on K(Ca)2 channels providing both selective activation and selective inhibition of the human K(Ca)2.1 subtype. |
PubMed:Direct condensation of sulfonamide and formamide: NaI-catalyzed synthesis of N-sulfonyl formamidine using TBHP as oxidant. |
PubMed:1,5,2,4,6,8-Dithiatetrazocine. Synthesis, computation, crystallography and voltammetry of the parent heterocycle. |
PubMed:Bioactivation of 4-Ipomeanol by a CYP4B enzyme in bovine lung and inhibition by HET0016. |
PubMed:Alkoxyamine-derived formamidines: configurational control and molecular folding. |
PubMed:Redetermination of (E)-N,N'-bis-(4-bromo-phen-yl)formamidine. |
PubMed:A new in vitro test to evaluate the resistance level against acaricides of the cattle tick, Rhipicephalus (Boophilus) microplus. |
PubMed:Inhibition of 20-HETE attenuates diabetes-induced decreases in retinal hemodynamics. |
PubMed:Modeling energy landscapes of proton motion in nonaqueous, tethered proton wires. |
PubMed:The cytochrome P450 4A/F-20-hydroxyeicosatetraenoic acid system: a regulator of endothelial precursor cells derived from human umbilical cord blood. |
PubMed:Microwave-assisted synthesis of a pyrazolyl ketone library for evaluation as p38 MAPK inhibitors in Werner syndrome cells. |
PubMed:Role of cytochrome P-450 metabolites in the regulation of renal function and blood pressure in 2-kidney 1-clip hypertensive rats. |
PubMed:Amine exchange in formamidines: an experimental and theoretical study. |
PubMed:20-Hydroxyeicosatetraenoic acid induces apoptosis in neonatal rat cardiomyocytes through mitochondrial-dependent pathways. |
PubMed:Synergy between fipronil and amitraz in a Rhipicephalus sanguineus tick residual contact test. |
PubMed:20-Hydroxyeicosatetraenoic acid synthesis is increased in human neutrophils and platelets by angiotensin II and endothelin-1. |
PubMed:Synthesis and crystal structure of a rare square-planar Co(II) complex of a hydroxyamidinate ligand. |
PubMed:Synthesis, X-ray crystallography characterization, vibrational spectroscopic, molecular electrostatic potential maps, thermodynamic properties studies of N,N'-di(p-thiazole)formamidine. |
PubMed:Selectivity of externally facing ion-binding sites in the Na/K pump to alkali metals and organic cations. |
PubMed:CYP4A2-induced hypertension is 20-hydroxyeicosatetraenoic acid- and angiotensin II-dependent. |
PubMed:Role of 20-hydroxyeicosatetraenoic and epoxyeicosatrienoic acids in the regulation of vascular function in a model of hypertension and endothelial dysfunction. |
PubMed:X-ray crystallography characterization, vibrational spectroscopy, NMR spectra and quantum chemical DFT/HF study of N,N'-di(2-methoxyphenyl)formamidine. |
PubMed:Discovery and characterization of an amidinotransferase involved in the modification of archaeal tRNA. |
PubMed:Double-stranded supramolecular assembly through salt bridge formation between rigid and flexible amidine and carboxylic acid strands. |
PubMed:A computational study of the nuclear magnetic resonance parameters for double proton exchange pathways in the formamide-formic acid and formamide-formamidine complexes. |
PubMed:The role of 20-hydroxyeicosatetraenoic acid in cerebral arteriolar constriction and the inhibitory effect of propofol. |
PubMed:Pharmacological characterization of a Bombyx mori alpha-adrenergic-like octopamine receptor stably expressed in a mammalian cell line. |
PubMed:Stereochemical and conformational exchanges in N,N'-di(2-pyridyl)formamidines: An X-ray and (1)H NMR study. |
PubMed:Down-regulation of 20-HETE synthesis and signaling inhibits renal adenocarcinoma cell proliferation and tumor growth. |
PubMed:Design, synthesis and pharmacological evaluation of a series of 5-carbethoxy-4-chloro-6-(substituted amino)pyrimidines as potential analgesic and anti-flammatory agents with very low ulcerogenic potential. |
PubMed:Expression and characterization of CYP4V2 as a fatty acid omega-hydroxylase. |
PubMed:Imidazol-2-ylidene-4-olate: an anionic N-heterocyclic carbene pre-programmed for further derivatization. |
PubMed:The role of 20-hydroxyeicosatetraenoic acid in adrenocorticotrophic hormone and dexamethasone-induced hypertension. |
PubMed:Cytotoxicity and cellular uptake of doxorubicin and its formamidine derivatives in HL60 sensitive and HL60/MX2 resistant cells. |
PubMed:Kidney androgen-regulated protein transgenic mice show hypertension and renal alterations mediated by oxidative stress. |
PubMed:Cytochrome P450 metabolites of arachidonic acid play a role in the enhanced cardiac dysfunction in diabetic rats following ischaemic reperfusion injury. |
PubMed:Role of 20-hydroxyeicosatetraenoic acid in altering vascular reactivity in diabetes. |
PubMed:Endothelin rather than 20-HETE contributes to loss of pial arteriolar dilation during focal cerebral ischemia with and without polymeric hemoglobin transfusion. |
PubMed:Cytotoxicity and inhibitory properties against topoisomerase II of doxorubicin and its formamidine derivatives. |
PubMed:Mechanisms of podocyte injury in diabetes: role of cytochrome P450 and NADPH oxidases. |
PubMed:Chronic blockade of 20-HETE synthesis reduces polycystic kidney disease in an orthologous rat model of ARPKD. |
PubMed:N,N-Bis(6-methyl-2-pyrid-yl)formamidine. |
PubMed:N-Ethyl-N-phenyl-N'-tosyl-formamidine. |
PubMed:N,N-Bis(2-pyrid-yl)formamidine. |
PubMed:N,N-Bis-(2,6-di-methyl-phen-yl)-N-hydroxyformamidine N,N'-bis-(2,6-dimethyl-phen-yl)-N-oxidoformamidinium dichloro-methane solvate. |
PubMed:Theoretical studies on the water-assisted hydrolysis of N,N-dimethyl-N'-(2',3'-dideoxy-3'-thiacytidine) formamidine with three water molecules. |
PubMed:Parallel synthesis of trisubstituted formamidines: a facile and versatile procedure. |
PubMed:Protective effect of 20-HETE analogues in experimental renal ischemia reperfusion injury. |
PubMed:Elevated production of 20-HETE in the cerebral vasculature contributes to severity of ischemic stroke and oxidative stress in spontaneously hypertensive rats. |
PubMed:The use of formamidine protection for the derivatization of aminobenzoic acids. |
PubMed:Role of CYP epoxygenases in A2A AR-mediated relaxation using A2A AR-null and wild-type mice. |
PubMed:Cytochrome P450 omega-hydroxylase inhibition reduces cardiomyocyte apoptosis via activation of ERK1/2 signaling in rat myocardial ischemia-reperfusion. |
PubMed:Intravenous formulation of N-hydroxy-N'-(4-n-butyl-2-methylphenyl)formamidine (HET0016) for inhibition of rat brain 20-hydroxyeicosatetraenoic acid formation. |
PubMed:A stable anionic N-heterocyclic carbene and its zwitterionic complexes. |
PubMed:Rapid and sensitive ultra-high-pressure liquid chromatography-quadrupole time-of-flight mass spectrometry for the quantification of amitraz and identification of its degradation products in fruits. |
PubMed:20-HETE mediates proliferation of renal epithelial cells in polycystic kidney disease. |
PubMed:Toward more efficient CCSD(T) calculations of intermolecular interactions in model hydrogen-bonded and stacked dimers. |
PubMed:Expression of CYP4A1 in U251 human glioma cell induces hyperproliferative phenotype in vitro and rapidly growing tumors in vivo. |
PubMed:Interaction of nitric oxide, 20-HETE, and EETs during functional hyperemia in whisker barrel cortex. |
PubMed:A facile preparation of imidazolinium chlorides. |
PubMed:Syntheses, structures and magnetism of linear tri- and tetra-copper chains containing anions of N,N'-bis(pyrimidine-2-yl)formamidine. |
PubMed:20-HETE increases renal sympathetic nerve activity via activation of chemically and mechanically sensitive muscle afferents. |
PubMed:Modulation of serum concentrations and hepatic metabolism of 17beta-estradiol and testosterone by amitraz in rats. |
PubMed:A monoclinic polymorph of N,N'-bis-(2,6-diisopropyl-phen-yl)formamidine. |
PubMed:Theoretical study on the hydrolysis mechanism of N,N-dimethyl-N'-(2-oxo-1, 2-dihydro-pyrimidinyl)formamidine: water-assisted mechanism and cluster-continuum model. |
PubMed:Hoogsteen vs. Watson-Crick base pairing: incorporation of 2-substituted adenine- and 7-deazaadenine 2'-deoxy-beta-D-ribonucleosides into oligonucleotides. |
PubMed:Synthesis of DNA-oligonucleotides damaged by arylamine-modified 2'-deoxyguanosine. |
PubMed:Facile synthesis of optically active imidazole derivatives. |
PubMed:Role of cytochrome P450 metabolites of arachidonic acid in regulation of corporal smooth muscle tone in diabetic and older rats. |
PubMed:Effect of acaricides on the activity of glutathione transferases from the parasitic mite Sarcoptes scabiei. |
PubMed:Steric modulation of coordination number and reactivity in the synthesis of lanthanoid(III) formamidinates. |
PubMed:Human enteric microsomal CYP4F enzymes O-demethylate the antiparasitic prodrug pafuramidine. |
PubMed:NMR studies of double proton transfer in hydrogen bonded cyclic N,N'-diarylformamidine dimers: conformational control, kinetic HH/HD/DD isotope effects and tunneling. |
PubMed:Crystal structures and solution behaviors of dinuclear d(10)-metal complexes containing anions of N,N'-bis(pyrimidine-2-yl)formamidine. |
PubMed:Adenine synthesis in interstellar space: mechanisms of prebiotic pyrimidine-ring formation of monocyclic HCN-pentamers. |
PubMed:A study on immunotoxicological effects of subacute amitraz exposure in rats. |
PubMed:Relative stability of formamidine and carbamate groups in the bifunctional pesticide formetanate hydrochloride. |
PubMed:Vascular cytochrome P450 4A expression and 20-hydroxyeicosatetraenoic acid synthesis contribute to endothelial dysfunction in androgen-induced hypertension. |
PubMed:Role of endogenous CYP450 metabolites of arachidonic acid in maintaining the glomerular protein permeability barrier. |
PubMed:Biological properties of new derivatives of daunorubicin. |
PubMed:Long-term fenofibrate treatment impairs endothelium-dependent dilation to acetylcholine by altering the cyclooxygenase pathway. |
PubMed:Cytochrome P-450 monooxygenases in control of renal haemodynamics and arterial pressure in anaesthetized rats. |
PubMed:Elevations in renal interstitial hydrostatic pressure and 20-hydroxyeicosatetraenoic acid contribute to pressure natriuresis. |
PubMed:Identification of pesticide transformation products in food by liquid chromatography/time-of-flight mass spectrometry via "fragmentation-degradation" relationships. |
PubMed:Synthesis and biological evaluation of some 5-ethoxycarbonyl-6-isopropylamino-4-(substitutedphenyl)aminopyrimidines as potent analgesic and anti-inflammatory agents. |
PubMed:Canine renal cortical necrosis and haemorrhage following ingestion of an Amitraz-formulated insecticide dip. |
PubMed:CYP4F enzymes are the major enzymes in human liver microsomes that catalyze the O-demethylation of the antiparasitic prodrug DB289 [2,5-bis(4-amidinophenyl)furan-bis-O-methylamidoxime]. |
PubMed:Nitric oxide/cytochrome P450 interactions in cyclosporin A-induced effects in the rat. |
PubMed:Synthesis and structural characterisation of heavy alkaline earth N,N'-bis(aryl)formamidinate complexes. |
PubMed:VEGF-induced relaxation of pulmonary arteries is mediated by endothelial cytochrome P-450 hydroxylase. |
PubMed:Increased renal vascular reactivity to ANG II after unilateral nephrectomy in the rat involves 20-HETE. |
PubMed:Comparison of the reproductive biology between acaricide-resistant and acaricide-susceptible Rhipicephalus (Boophilus) microplus (Acari: Ixodidae). |
PubMed:Protective effect of the 20-HETE inhibitor HET0016 on brain damage after temporary focal ischemia. |
PubMed:An efficient synthesis of acyclic N7- and N9-adenine nucleosides via alkylation with secondary carbon electrophiles to introduce versatile functional groups at the C-1 position of acyclic moiety. |
PubMed:Glial cells dilate and constrict blood vessels: a mechanism of neurovascular coupling. |
PubMed:Acute amitraz poisoning in adults: clinical features, laboratory findings, and management. |
PubMed:9L gliosarcoma cell proliferation and tumor growth in rats are suppressed by N-hydroxy-N'-(4-butyl-2-methylphenol) formamidine (HET0016), a selective inhibitor of CYP4A. |
PubMed:Synthesis and in solution and solid state structural study of intramolecular Pt...H interactions in pentafluorophenyl platinum(II) complexes containing the ligands triazene, formamidine, and 2-aminopyridine. |
PubMed:Amitraz: an unusual aetiology of Ogilvie's syndrome. |
PubMed:Taking the 20-HETE out of the cardiovascular system: the potential of 20-HETE synthesis inhibitors. |
PubMed:Cytochrome P450 4A isoform inhibitory profile of N-hydroxy-N'-(4-butyl-2-methylphenyl)-formamidine (HET0016), a selective inhibitor of 20-HETE synthesis. |
PubMed:Human U251 glioma cell proliferation is suppressed by HET0016 [N-hydroxy-N'-(4-butyl-2-methylphenyl)formamidine], a selective inhibitor of CYP4A. |
PubMed:Stable planar six-pi-electron six-membered N-heterocyclic carbenes with tunable electronic properties. |
PubMed:Inhibition of Ca2+/calmodulin-dependent protein kinase II, RAS-GTPase and 20-hydroxyeicosatetraenoic acid attenuates the development of diabetes-induced vascular dysfunction in the rat carotid artery. |
PubMed:Elevated plasma cysteinylglycine levels caused by cilastatin-associated antibiotic treatment. |
PubMed:Structural and magnetic evidence concerning spin crossover in formamidinate compounds with ru2 5+ cores. |
PubMed:Steric engineering of C-F activation with lanthanoid formamidinates. |
PubMed:A theoretical study on the mechanism of the reductive half-reaction of xanthine oxidase. |
PubMed:Linear and cyclic tetranuclear copper(I) complexes containing anions of N,N'-bis(pyrimidine-2-yl)formamidine. |
PubMed:Inhibitors of cytochrome P450 4A suppress angiogenic responses. |
PubMed:Paramagnetic precursors for supramolecular assemblies: selective syntheses, crystal structures, and electrochemical and magnetic properties of Ru2(O2CMe)4-n(formamidinate)nCl complexes, n = 1-4. |
PubMed:An in vitro larval immersion microassay for identifying and characterizing candidate acaricides. |
PubMed:Interactions of novel morpholine and hexamethylene derivatives of anthracycline antibiotics with DNA. |
PubMed:Modular synthesis of formamidines and their formation of stable organogels. |
PubMed:Reaction products of W(CO)(6) with formamidines; electronic structure of a W(2)(mu-CO)(2) core with unsymmetric bridging carbonyls. |
PubMed:Effects of amitraz on cytochrome P450-dependent monooxygenases and estrogenic activity in MCF-7 human breast cancer cells and immature female rats. |
PubMed:[Control strategies against Varroa mites]. |
PubMed:Amitraz poisoning: clinical and laboratory findings. |
PubMed:Experimental and theoretical evidence of basic site preference in polyfunctional superbasic amidinazine: N(1),N(1)-dimethyl-N(2)-beta-(2-pyridylethyl)formamidine. |
PubMed:Detection and characterization of amitraz resistance in the southern cattle tick, Boophilus microplus (Acari: Ixodidae). |
PubMed:Potent nonclassical nucleoside antiviral drugs based on the N,N-diarylformamidine concept. |
PubMed:Expanded chemistry of formamidine ureas. |
PubMed:Formamidine ureas as tunable electrophiles. |
PubMed:Smooth muscle--specific expression of CYP4A1 induces endothelial sprouting in renal arterial microvessels. |
PubMed:Molecular squares with paramagnetic diruthenium corners: synthetic and crystallographic challenges. |
PubMed:Inhibitors of 20-HETE formation promote salt-sensitive hypertension in rats. |
PubMed:First practical synthesis of formamidine ureas and derivatives. |
PubMed:Report of eight children with amitraz intoxication. |
PubMed:Contribution of 5-hydroxytryptamine1B receptors and 20-hydroxyeiscosatetraenoic acid to fall in cerebral blood flow after subarachnoid hemorrhage. |
PubMed:Contributions of 20-HETE to the antihypertensive effects of Tempol in Dahl salt-sensitive rats. |
PubMed:Structural studies of N,N'-di(ortho-fluorophenyl)formamidine group 1 metallation. |
PubMed:CYP4A metabolites of arachidonic acid and VEGF are mediators of skeletal muscle angiogenesis. |
PubMed:NMR studies of the tautomerism of cyclo-tris(4-R-2,6-pyridylformamidine) in solution and in the solid state. |
PubMed:Comparative toxic and genotoxic effects of chloroacetanilides, formamidines and their degradation products on Vibrio fischeri and Chironomus riparius. |
PubMed:Synthesis of 99mTc-ciprofloxacin by different methods and its biodistribution. |
PubMed:Basic toxicological approach has been effective in two poisoned patients with amitraz ingestion: case reports. |
PubMed:20-HETE contributes to the acute fall in cerebral blood flow after subarachnoid hemorrhage in the rat. |
PubMed:[Effects of occupational exposure to formamidines on cardiovascular functions]. |
PubMed:Discovery of a N'-hydroxyphenylformamidine derivative HET0016 as a potent and selective 20-HETE synthase inhibitor. |
PubMed:Quadruply Bonded Dichromium Complexes with Variously Fluorinated Formamidinate Ligands. |
PubMed:"One-pot" synthesis and antimalarial activity of formamidine derivatives of 4-anilinoquinoline. |
PubMed:Role of guanylyl cyclase and cytochrome P-450 on renal response to nitric oxide. |
PubMed:Minimal amidine structure for inhibition of nitric oxide biosynthesis. |
PubMed:HET0016, a potent and selective inhibitor of 20-HETE synthesizing enzyme. |
PubMed:Proton motion and proton transfer in the formamidine-formic acid complex: an Ab initio projector augmented wave molecular dynamics study. |
PubMed:Interaction of formamidine pesticides with the presynaptic alpha(2)-adrenoceptor regulating. |
PubMed:Dinuclear and heteropolynuclear complexes containing Mo2(4+) units. |
PubMed:Tyramine injections reduce locust viability. |
PubMed:The ability of new formamidine sugar-modified derivatives of daunorubicin to stimulate free radical formation in three enzymatic systems: NADH dehydrogenase, NADPH cytochrome P450 reductase and xanthine oxidase. |
PubMed:Susceptibility to two pyrethroids in Boophilus microplus (Acari: Ixodidae) populations of northwest Argentina. Preliminary results. |
PubMed:Effects of the pesticide amitraz and its metabolite BTS 27271 on insulin and glucagon secretion from the perfused rat pancreas: involvement of alpha2D-adrenergic receptors. |
PubMed:In vitro and in vivo effects of formamidines in locust (Locusta migratoria migratorioides). |
PubMed:Lorentzian noise in single gramicidin A channel formamidinium currents. |
PubMed:Isolation of a cDNA for an octopamine-like, G-protein coupled receptor from the cattle tick, Boophilus microplus. |
PubMed:Neuroendocrine and reproductive effects of contemporary-use pesticides. |
PubMed:S-oxygenation of thiourea results in the formation of genotoxic products. |
PubMed:The effect of biogenic amines and their analogs on carbohydrate metabolism in the fat body of the cockroach Blaberus discoidalis. |
PubMed:An unusual poisoning with the unusual pesticide amitraz. |
PubMed:Molecular dynamics study of free energy profiles for organic cations in gramicidin A channels. |
PubMed:Synthesis and assessment of formamidines as new histamine H2-receptor antagonists. |
PubMed:Novel histamine H3 receptor antagonists: synthesis and evaluation of formamidine and S-methylisothiourea derivatives. |
PubMed:Synergism of toxicity of N,N-diethyl-m-toluamide to German cockroaches (Orthoptera: Blattellidae) by hydrolytic enzyme inhibitors. |
PubMed:Evaluation of C-(beta-D-galactosyl) and C-(2-deoxy-D-lyxo-hex-1-enopyranosyl) (D-galactal type) derivatives as inhibitors of beta-D-galactosidase from Escherichia coli. |
PubMed:Novel Bicyclic Lactams as XaaPro Type VI beta Turn Mimics: Design, Synthesis, and Evaluation. |
PubMed:Total Synthesis of (-)-Tetrahydropalmatine via Chiral Formamidine Carbanions: Unexpected Behavior with Certain Ortho-Substituted Electrophiles. |
PubMed:Synthesis and Structural Studies of Platinum Complexes Containing Monodentate, Bridging, and Chelating Formamidine Ligands. |
PubMed:The permeation of organic cations through cAMP-gated channels in mammalian olfactory receptor neurons. |
PubMed:Gramicidin tryptophans mediate formamidinium-induced channel stabilization. |
PubMed:Inhibition of insulin release by a formamidine pesticide amitraz and its metabolites in a rat beta-cell line: an action mediated by alpha-2 adrenoceptors, a GTP-binding protein and a decrease in cyclic AMP. |
PubMed:Influence of the formamidine pesticide amitraz and its metabolites on porcine myometrial contractility: involvement of alpha 2-adrenoceptors and Ca2+ channels. |
PubMed:Monovalent amidiniums block calcium channels in chick sensory neurons. |
PubMed:Antinociceptive effect of amitraz in mice and rats. |
PubMed:N4-(dialkylamino)methylene derivatives of 2'-deoxycytidine and arabinocytidine: physicochemical studies for potential prodrug applications. |
PubMed:Properties of an arylalkylamine N-acetyltransferase from the nematode, Ascaridia galli. |
PubMed:Formamidinium-induced dimer stabilization and flicker block behavior in homo- and heterodimer channels formed by gramicidin A and N-acetyl gramicidin A. |
PubMed:Amides and formamidines with antinociceptive activity (note II). |
PubMed:Amides and formamidines with antinociceptive activity (note I). |
PubMed:Influence of the formamidine pesticide chlordimeform on ovulation in the female hamster: dissociable shifts in the luteinizing hormone surge and oocyte release. |
PubMed:Effects of amitraz on motor function. |
PubMed:The permeation properties of small organic cations in gramicidin A channels. |
PubMed:Calcium entry blockade as a mechanism for chlordimeform-induced inhibition of motor activity in the isolated guinea-pig ileum. |
PubMed:Gramicidin channel selectivity. Molecular mechanics calculations for formamidinium, guanidinium, and acetamidinium. |
PubMed:Comet Halley as an aggregate of interstellar dust and further evidence for the photochemical formation of organics in the interstellar medium. |
PubMed:Sublethal effects of the formamidine amitraz on honeybees gut lipids, following in vivo injections. |
PubMed:Estimation of flavin-containing monooxygenase activities in crude tissue preparations by thiourea-dependent oxidation of thiocholine. |
PubMed:The formamidine pesticides chlordimeform and amitraz decrease hepatic glutathione in mice through an interaction with alpha 2-adrenoceptors. |
PubMed:Adenine photodimerization in deoxyadenylate sequences: elucidation of the mechanism through structural studies of a major d(ApA) photoproduct. |
PubMed:Substituent effect on the stereochemistry of H2-receptor antagonists of the phenylformamidine series. A conformation-dependent mode of interaction with the H2 receptor. |
PubMed:Rat strain and stock comparisons using a functional observational battery: baseline values and effects of amitraz. |
PubMed:Interaction between amitraz and alpha 2-adrenoceptors inhibits epinephrine-induced canine platelet aggregation. |
PubMed:Quantification of imipenem's primary metabolite in plasma by postcolumn chemical rearrangement and UV detection. |
PubMed:Synthesis and biological activity of the 2-desamino and 2-desamino-2-methyl analogues of aminopterin and methotrexate. |
PubMed:Formamidines as synergists of cypermethrin in susceptible and pyrethroid resistant house flies (Diptera: Muscidae). |
PubMed:Prebiotic synthesis of histidine. |
PubMed:Synthesis and biological evaluation of new antimuscarinic compounds with amidine basic centers. A useful bioisosteric replacement of classical cationic heads. |
PubMed:Hexocyclium derivatives with a high selectivity for smooth muscle muscarinic receptors. |
PubMed:[Production and antineoplastic activity of new asymmetric azines on the rubomycin base]. |
PubMed:Irreversible H2-antagonism of the four isomeric butyl analogues of mifentidine. |
PubMed:[The effect of pesticides-CDM and AMZ on inhibition of the binding of 3H-clonidine to alpha 2-adrenoreceptor in rat forebrain tissue]. |
PubMed:Central and peripheral alpha-adrenoceptor actions of amitraz in the dog. |
PubMed:Synthesis and structure-activity relationship of C5-substituted analogues of (+-)-10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5,10-imine [(+-)-desmethyl-MK801]: ligands for the NMDA receptor-coupled phencyclidine binding site. |
PubMed:Octopamine uptake and metabolism in the insect nervous system. |
PubMed:Synthesis of 11C-labeled (+-)-5-methyl-10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5,10-imin e [(+-)-[11C]MK801]. |
PubMed:Amitraz-induced glucose intolerance in rats: antagonism by yohimbine but not by prazosin. |
PubMed:Formamidine pesticides and alpha 2-adrenoceptors: studies with amitraz and chlordimeform in rats and development of a radioreceptor binding assay. |
PubMed:The formamidine amitraz as a hyperglycemic alpha-agonist in worker honeybees (Apis mellifera mellifera L.) in vivo. |
PubMed:N-(fluoroethyl)(imidazolylphenyl)formamidines. The issue of the active species of mifentidine. |
PubMed:Acute and chronic effects of the pesticide amitraz on alpha 2-adrenoceptors in mouse brain. |
PubMed:Investigations of amitraz neurotoxicity in rats. III. Effects on motor activity and inhibition of monoamine oxidase. |
PubMed:Technetium-99m spiperone dithiocarbamate: a potential radiopharmaceutical for dopamine receptor imaging with SPECT. |
PubMed:Enhanced susceptibility to kindling by chlordimeform may be mediated by a local anesthetic action. |
PubMed:Comparison of chlordimeform and carbaryl using a functional observational battery. |
PubMed:Permeability to various cations of the voltage-dependent sodium channel of isolated rat hippocampal pyramidal neurons. |
PubMed:Increased hippocampal excitability produced by amitraz. |
PubMed:Formamidine pesticides enhance susceptibility to kindled seizures in amygdala and hippocampus of the rat. |
PubMed:Alpha 2-adrenoceptors as a target for formamidine pesticides: in vitro and in vivo studies in mice. |
PubMed:Effects of topical application of amitraz on plasma glucose and insulin concentrations in dogs. |
PubMed:The toxicity of disulphides to isolated hepatocytes and mitochondria. |
PubMed:The bradycardic and mydriatic effects of chlordimeform and its demethylated analogs in the rat: antagonism by idazoxan but not by prazosin. |
PubMed:Characterization of nonheme iron and reaction mechanism of bromoperoxidase in Corallina pilulifera. |
PubMed:Investigations of amitraz neurotoxicity in rats. I. Effects on operant performance. |
PubMed:Investigations of amitraz neurotoxicity in rats. II. Effects on visual evoked potentials. |
PubMed:Cardiovascular and respiratory effects of the acaricide amitraz. |
PubMed:Further evidence to support the alpha 2-adrenergic nature of amitraz-induced decrease in intestinal motility. |
PubMed:Interaction of the pesticide chlordimeform with adrenergic receptors in mouse brain: an in vitro study. |
PubMed:Cholinergic involvement in the action of formetanate on operant behavior in rats. |
PubMed:Mechanism of ammonium translocation in rat liver mitochondria. Finger-printing of the translocator. |
PubMed:Prebiotic synthesis of imidazole-4-acetaldehyde and histidine. |
PubMed:Technetium-99m diethyldithiocarbamate (DDC): comparison with thallium-201 DDC as an agent for brain imaging. |
PubMed:Differential effects of formamidine pesticides on fixed-interval behavior in rats. |
PubMed:The analgesic activity of a clonidine analog. The formamidine, U-47,476A. |
PubMed:Induction of hepatic drug-metabolising enzymes following treatment of rats and mice with chlordimeform. |
PubMed:Yohimbine attenuates the delayed lethality induced in mice by amitraz, a formamidine pesticide. |
PubMed:Thermoregulation in mice following acute chlordimeform administration. |
PubMed:Monoamine oxidase inhibition cannot account for changes in visual evoked potentials produced by chlordimeform. |
PubMed:Interactions of permeant cations with sodium channels of squid axon membranes. |
PubMed:Receptors for 3H-octopamine in the adult firefly light organ. |
PubMed:Body temperature-dependent and independent actions of chlordimeform on visual evoked potentials and axonal transport in optic system of rat. |
PubMed:The preparation of carbon-11 labelled proline for positron emission tomography. Preliminary distribution studies in rats with Walker 256 carcinosarcoma. |
PubMed:Effects of chlordimeform on cardiovascular functional parameters: Part 1. Lethality and arrhythmogenicity in the geriatric rat. |
PubMed:Suppression of the antibody response by a formamidine pesticide: dependence on the route of exposure. |
PubMed:Formamidine-mediated inhibition of rat platelet aggregation. |
PubMed:Mifentidine: evaluation of antiandrogen effects and kidney function studies. |
PubMed:Conformational studies of two histamine H2-receptor antagonistic phenylformamidines: mifentidine and its guanidinothiazole analogue DA 4643. |
PubMed:Chlordimeform produces profound, selective, and transient changes in visual evoked potentials of hooded rats. |
PubMed:The pharmacokinetics of imipenem (thienamycin-formamidine) and the renal dehydropeptidase inhibitor cilastatin sodium in normal subjects and patients with renal failure. |
PubMed:Effect of amitraz and chlordimeform on heart rate and pupil diameter in rats: mediated by alpha 2-adrenoreceptors. |
PubMed:(Imidazolylphenyl)formamidines. A structurally novel class of potent histamine H2 receptor antagonists. |
PubMed:Relaxation of rabbit aorta by chlordimeform. |
PubMed:Hot atoms in cosmic chemistry. |
PubMed:Metabolism of four thiobis(formamidine) insecticides in the mouse and the rat. |
PubMed:Some effects of the formamidine pesticide chlordimeform on the behavior of mice. |
PubMed:Permeability to various cations of the voltage-dependent sodium channel of rat single heart cells. |
PubMed:5-Hydroxytryptamine stimulates fluid secretion in locust malpighian tubules independently of cAMP. |
PubMed:Extrapolation from safety data to management of poisoning with reference to amitraz (a formamidine pesticide) and xylene. |
PubMed:Animal studies on the treatment of poisoning by amitraz (a formamidine pesticide) and xylene. |
PubMed:A randomized study comparing clinical efficacy and safety of thienamycin formamidine (MK0787)/renal dipeptidase inhibitor (MK0791) and cefazolin. |
PubMed:Northienamycin and 8-epi-thienamycin, new carbapenems from Streptomyces cattleya. |
PubMed:Experimental studies of drug-induced impaction colic in the horse. |
PubMed:Potential neuromuscular toxicity of N'-(2,4-xylyl)-N-methyl formamidine HCl in rodents. |
PubMed:Perturbation of hydrogen bonds in the adenine . thymine base pair by Na+: A quantum chemical study. |
PubMed:Synthesis of N'-aryl-N3-(substituted)-alpha, alpha'-thio-bis-formamidine dihydrochlorides and their effect on blood sugar level of albino rats. |
PubMed:Effects of Selected Insecticides and Nematicides on the In Vitro Development of the Entomogenous Nematode Neoaplectana carpocapsae. |
PubMed:Interaction of formamidines with the platelet 5-hydroxytryptamine uptake system. |
PubMed:The influence of reducing agents on the composition of 99Tc-complexes: implications for 99mTc-radiopharmaceutical preparation. |
PubMed:Effect of amitraz on contractions of the guinea-pig ileum in vitro. |
PubMed:Reduction of aspirin-induced ulcers by a new imidazoline anti-inflammatory agent. |
PubMed:Inhibition of rat platelet 5-hydroxytryptamine uptake by chlordimeform. |
PubMed:Transport of ammonium and methylammonium ions by Azotobacter vinelandii. |
PubMed:Response of adrenal catecholamine to a newly synthesized chemical radioprotector. |
PubMed:Excretion balance, metabolic fate and tissue residues following treatment of rats with amitraz and N'-(2,4-dimethylphenyl)-N-methylformamidine. |
PubMed:The use of formamidine sulphinic acid in the preparation of 99mTc-labelled radiopharmaceuticals--a cautionary note. |
PubMed:Action of formamidine pesticides on octopamine receptors. |
PubMed:Pharmacological modulation of edema mediated by prostaglandin, serotonin and histamine. |
PubMed:Trial of a new compound as a chemical radioprotector and its effect on melatonin. |
PubMed:Anti-inflammatory and analgesic profile of amidines of 3-amino-1,2,4-benzotriazine and 3-amino-1,2,4-benzotriazine-1-oxide. |
PubMed:The effects of U-40481, demethylchlordimeform, and formetanate on calcium flux in the isolated rabbit aorta. |
PubMed:Formamidine pesticides: octopamine-like actions in a firefly. |
PubMed:A survey of reducing agents for the synthesis of tetraphenylarsonium oxotechnetiumbis(ethanedithiolate) from [99Tc] pertechnetate in aqueous solution. |
PubMed:Preparation of technetium-99m glucoheptonate utilizing formamidine sulfinic acid. |
PubMed:Cation selectivity of acetylcholine-activated ionic channel of frog endplate. |
PubMed:Thiourea and cyanamide as inhibitors of thyroid peroxidase: the role of iodide. |
PubMed:Mode of action of formamidine pesticides: an evaluation of monoamine oxidase as the target. |
PubMed:Prostaglandin synthesis inhibited by formamidine pesticides. |
PubMed:Increased feeding in rats treated with chlordimeform and related formamidines: a new class of appetite stimulants. |
PubMed:Evaluation of formamidine sulfinic acid and other reducing agents for use in the preparation of Tc-99m labeled radiopharmaceuticals. |
PubMed:Formamidine acaricides. Toxicity and metabolism studies with twospotted spider mites, Tetranychus urticae Koch. |
PubMed:Cation permeability ratios of sodium channels in normal and grayanotoxin-treated squid axon membranes. |
PubMed:Permeability of the sodium channel in Myxicola to organic cations. |
PubMed:Chemistry and toxicology of quinoxaline, organotin, organofluorine, and formamidine acaricides. |
PubMed:Chemistry, biological activity, and uses of formamidine pesticides. |
PubMed:Formamidine acaricides: toxicological studies with the cattle tick. |
PubMed:Studies on models for tetrahydrofolic acid. V.A. kinetically significant transport process in general base catalyzed aminolysis of a formamidine. |
PubMed:Toxicity to Boophilus microplus of formamidine acaricides and related compounds, and modification of toxicity by certain insecticide synergists. |
PubMed:[Inhibition of serum transamidinase by formamidine disulfide: identification of the SH-group in the active center of the enzyme]. |
PubMed:The permeability of the sodium channel to organic cations in myelinated nerve. |
PubMed:[Formamidine derivatives of anthelmintic effect. (Preliminary report)]. |
PubMed:On the pharmacological characteristic of some pyridine derivatives of formamidine and the relationship of their structure and action. |
PubMed:Pharmacological assaying of some compounds of the formamidine group. |
PubMed:FORMAMIDINE SULFINIC ACID AS A BIOCHEMICAL REDUCING AGENT. |
PubMed:Formamidine group transfer in extracts of human pancreas, liver, and kidney. |
PubMed:Inhibition of sulfhydryl enzymes by formamidine disulfide. |
PubMed:The reaction of ketones with formamidine disulfide. |
PubMed:Oxidation-reduction potentials of thiol-dithio systems: thiourea-formamidine disulfide. |
PubMed:Synthesis of 4-hydroxyquinolines; a modified preparation through bis-(m-chlorophenyl)-formamidine. |